Reference: Exelixis drugs,targets & Indications
Drug,Target,Status,Indication
XL119* Topoisomerase 2 Phase III Biliary Tract Cancer
XL999** VEGFR2, PDGFR,FGFR, FLT3 Phase II Renal Cell Carcinoma, Colon, Ovarian,NSCLC, AML, Multiple Myeloma
XL647** VEGFR2, EGFR,HER2 Phase II NSCLC
XL784** ADAM10, MMP-2 Phase II Diabetic Nephropathy
XL880 c-MET, VEGFR2 Phase II Papillary Cell Carcinoma
XL820 c-KIT, VEGFR2,PDGFR Phase I Solid Tumors
XL844 CHK1, CHK2 Phase I Solid Tumors, Hematologic Malignancies
XL184 c-MET, VEGFR2 Phase I Solid Tumors
XL228 ABL, IGF1R, SRC IND Filed Solid Tumors, Hematologic Malignancies
XL281 RAF IND Filed Solid Tumors
XL418 AKT, S6K Preclinical Solid Tumors
XL518 MEK Preclinical Solid Tumors
XL765 PI-3K, mTOR Preclinical Solid Tumors
XL147 PI-3K Preclinical Solid Tumors
XL019 JAK2 Preclinical Myeloid/Lymphoid Malignancies
XL550*** Mineralocorticoid Receptor Preclinical Hypertension
XL335*** Farsenoid Receptor Preclinical Atherosclerosis
EXEL2255*** Liver X Receptor Preclinical Atherosclerosis |